Product Name CAS NO. System support Document support Classification
(1S)-1,5-Anhydro-1-C-[3-[[5-(4-fluorophenyl)-2-thienyl]methyl]-4-methylphenyl]-D-glucitol tetraacetate 866607-35-4 ISO/ GMP TDP/DMF Canagliflozin hemihydrate
2-(4-Fluorophenyl)-5-[(5-iodo-2-methylphenyl)methyl]thiophene 898566-17-1 ISO/ GMP TDP Canagliflozin hemihydrate
Dapagliflozin base 461432-26-8 ISO/ GMP TDP/DMF Dapagliflozin propanediol monohydrate
(1S)-1,5-Anhydro-1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-D-glucitol tetraacetate 461432-25-7  ISO/ GMP TDP/DMF Dapagliflozin propanediol monohydrate
Methyl 1-C-[4-chloro-3-(4-ethoxybenzyl)phenyl]-α-D-glucopyranoside 714269-57-5 ISO TDP Dapagliflozin propanediol monohydrate
5-bromo-2-chloro-4’-ethoxydiphenylmethane 461432-23-5 ISO TDP Dapagliflozin propanediol monohydrate
(5-Bromo-2-chlorophenyl)(4-ethoxyphenyl)methanone 461432-22-4 ISO TDP Dapagliflozin propanediol monohydrate
5-iodo-2-chloro-4'-ethoxydiphenylmethane 1103738-29-9 ISO TDP Dapagliflozin propanediol monohydrate
5-Bromo-2-chlorobenzoic acid 21739-92-4 ISO TDP Dapagliflozin propanediol monohydrate
(1S)-1,5-Anhydro-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methyl]phenyl]-D-glucitol tetraacetate 915095-99-7 ISO/ GMP TDP/DMF Empagliflozin
Methyl 1-C-[4-chloro-3-[[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methyl]phenyl]-alpha-D-glucopyranoside 1279691-36-9 ISO TDP Empagliflozin
(3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan 915095-89-5 ISO TDP Empagliflozin
(3S)-3-[4-[(5-iodo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan 915095-94-2 ISO TDP Empagliflozin
(2-Chloro-5-iodophenyl)[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methanone 915095-87-3 ISO TDP Empagliflozin
2,3,4,6-Tetrakis-O-trimethylsilyl-D-gluconolactone 32384-65-9 ISO TDP Empagliflozin
(S)-(+)-3-Hydroxytetrahydrofuran 86087-23-2 ISO TDP Empagliflozin
Methyl (5S)-5-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-thio-beta-L-xylopyranoside 2,3,4-triacetate 1018899-03-0 ISO/ GMP TDP/DMF Sotagliflozin
(4-Chloro-3-(4-ethoxybenzyl)phenyl)((3aS,5R,6S,6aS)-6-hydroxy-2,2-dimethyltetrahydrofuro[2,3-d][1,3]dioxol-5-yl)methanone 1103738-30-2 ISO TDP Sotagliflozin
(5S)-4,5-O-(1-Methylethylidene)-1-C-4-morpholinyl-D-xylo-pentodialdo-5,2-furanose 1103738-19-7 ISO TDP Sotagliflozin
Ipragliflozin 761423-87-4 ISO/ GMP TDP/DMF Ipragliflozin
(1S)-1,5-Anhydro-1-C-[3-(benzo[b]thien-2-ylmethyl)-4-fluorophenyl]-D-glucitol 2,3,4,6-tetraacetate 1034305-21-9 ISO/ GMP TDP/DMF Ipragliflozin
2-(5-Bromo-2-fluorobenzyl)benzo[b]thiophene 1034305-17-3 ISO TDP Ipragliflozin
(2S,3R,4S,5S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6,6-bis(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol 1528636-39-6 ISO TDP Ertugliflozin
(S)-2-((2-Oxo-3-(4-(3-oxomorpholino)phenyl)oxazolidin-5-yl)methyl)isoindoline-1,3-dione 446292-08-6 ISO TDP Rivaroxaban
(S)-4-(4-(5-(Aminomethyl)-2-oxooxazolidin-3-yl)phenyl)morpholin-3-one.HCl 898543-06-1 ISO TDP Rivaroxaban
2-[(2R)-2-Hydroxy-3-[[4-(3-oxo-4-morpholinyl)phenyl]amino]propyl]-1H-isoindole-1,3(2H)-dione 446292-07-5 ISO TDP Rivaroxaban
(S)-(+)-N-(2,3-Epoxypropyl)phthalimide 161596-47-0 ISO TDP Rivaroxaban
4-(4-aminophenyl)morpholin-3-one 438056-69-0 ISO TDP Rivaroxaban
5-Chloro-2-thiophenecarboxylic acid 24065-33-6  ISO TDP Rivaroxaban
Benzeneazomalononitrile 6017-21-6 ISO TDP Riociguat
Pyrazolo[3,4-b]pyridine-3-carboximidamide,1-[(2-fluorophenyl)methyl]-, monohydrochloride 256499-19-1 ISO TDP Riociguat
5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carbonitrile 1350653-26-7 ISO TDP Vericiguat
4-Chloro-7-tosyl-7H-pyrrolo[2,3-d]pyrimidine 479633-63-1 ISO TDP Tofacitinib
4-chloro-7H-pyrrolo[2,3-d]pyriMidine 3680-69-1 ISO TDP Tofacitinib
Pyrrolo[2,3-d]pyrimidin-4-ol 3680-71-5 ISO TDP Tofacitinib
2-[1-(Ethylsulfonyl)-3-azetidinylidene]acetonitrile 1187595-85-2 ISO TDP Baricitinib
tert-butyl 4-chloro-7H-pyrrolo[2,3-d]pyrimidine-7-carboxylate 1236033-21-8 ISO TDP Baricitinib
Abrocitinib 1622902-68-4 ISO TDP Abrocitinib
benzyl ((1s,3s)-3-(methylamino)cyclobutyl)carbamate hydrochloride 2204290-99-1 ISO TDP Abrocitinib
N-(5-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide 1142943-96-1 ISO TDP Filgotinib
4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)thiomorpholine 1,1-dioxide 1092563-25-1 ISO TDP Filgotinib
(4-Chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methylpivalate 1146629-75-5 ISO TDP Ruxolitinib
1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 1029716-44-6 ISO TDP Ruxolitinib
3-Cyclopentyl-acrylonitrile 591769-05-0 ISO TDP Ruxolitinib
benzyl (2S,5R)-5-amino-2-methylpiperidine-1-carboxylate hydrogen chloride 1207853-23-3 ISO TDP Ritlecitinib
(S)-1-(2,6-Dichloro-3-fluorophenyl)ethanol 877397-65-4 ISO TDP Crizotinib
(R)-5-broMo-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)pyridin-2-aMine 877399-00-3 ISO TDP Crizotinib
tert-Butyl 4-[4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]piperidine-1-carboxylate 877399-74-1 ISO TDP Crizotinib
(R)-2-(2,5-difluorophenyl)pyrrolidine (R)-2-hydroxysuccinate 1919868-77-1 ISO TDP Larotrectinib
(S)-pyrrolidin-3-ol 100243-39-8 ISO TDP Larotrectinib
(S)-1-(5-fluoro-2-iodophenyl)ethan-1-ol 1454847-96-1 ISO TDP Lorlatinib
(R)-pyrrolidin-3-ol 2799-21-5 ISO TDP Asciminib
4-(Chlorodifluoromethoxy)aniline 39065-95-7 ISO TDP Asciminib
5-Chloro-2-((R)-5-Methyl-[1,4]diazepan-1-yl)benzooxazole hydrochloride 1266664-66-7 ISO TDP Suvorexant
4-((2-aminoethyl)(5-chlorobenzo[d]oxazol-2-yl)amino)butan-2-onedimethanesulfonate 1276666-12-6 ISO TDP Suvorexant
(R)-1-benzyl-5-methyl-1,4-diazepane 1620097-06-4 ISO TDP Suvorexant
5-Methyl-2-(2H-1,2,3-triazol-2-yl)benzoicacid 956317-36-5 ISO TDP Suvorexant
5-bromo-2-(2-methyl-2H-tetrazol-5-yl)pyridine 380380-64-3 ISO TDP Tedizolid
1H-IMidazole, 5,5'-[1,1'-biphenyl]-4,4'-diylbis[2-(2S)-2-pyrrolidinyl-, hydrochloride (1:4) 1009119-83-8 ISO TDP Tedizolid
(R)-3-(4-bromo-3-fluorophenyl)-5-(hydroxymethyl)oxazolidin-2-one 444335-16-4 ISO TDP Tedizolid
Torezolid  856866-72-3 ISO TDP Tedizolid
(5S,6S,9R)-5-Amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-ol dihydrochloride 1373116-07-4 ISO TDP Rimegepant sulfate
(9R)-9-hydroxy-6,7,8,9-tetrahydrocyclohepta[b]pyridin-5-one 1190363-44-0 ISO TDP Rimegepant sulfate
1-(1-(1H-imidazole-1-carbonyl)piperidin-4-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one 1373116-06-3 ISO TDP Rimegepant sulfate
2-Oxo-1-(4-piperidinyl)-2,3-dihydro-1H-imidazo[4,5-b]pyridine dihydrochloride 781649-84-1 ISO TDP Rimegepant sulfate
3-(piperidin-4-yl)quinolin-2(1h)-one hydrochloride 855778-84-6 ISO TDP Zevagepant
methyl (2R)-2-amino-3-(7-methyl-1H-indazol-5-yl)propanoate dihydrochloride 1414976-14-9 ISO TDP Zevagepant
1-(1-Methyl-4-piperidinyl)piperazine 23995-88-2 ISO TDP Zevagepant
2-Chloropyridine-3-sulfonyl chloride 6684-06-6 ISO TDP Zibotentan
isobutyl 3-Methoxy-5-Methylpyrazin-2-ylcarbaMate 186497-47-2 ISO TDP Zibotentan
[4-(1,3,4-oxadiazol-2-yl)phenyl]boronic acid 276694-22-5 ISO TDP Zibotentan
1-isopropylpyrimidine-2,4,6(1H,3H,5H)-trione 69998-14-7 ISO TDP Mavacamten
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